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CBPD-268

Product Specifications

Target

PROTACs|||Histone Acetyltransferase

Related Pathways

Chromatin/Epigenetic|||PROTAC

Bioactivity

CBPD-268 is an effective orally active CBP/p300 PROTAC degrader, with a DC50 value of ? 0.03 nM. It induces degradation of CBP/p300 and inhibits cell growth, exhibiting antitumor activity. Additionally, CBPD-268 shows potential for research in AR-positive prostate cancer.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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