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YCH2823

Product Specifications

Target

Apoptosis, DUB

Related Pathways

Cell Cycle/Checkpoint, Apoptosis, DNA Damage/DNA Repair, Ubiquitination

Bioactivity

YCH2823 is an inhibitor of USP7 (IC50= 49.6 nM; Kd= 0.117 μM) and demonstrates significant efficacy in suppressing both wild-type TP53 tumors and mutated tumors. It is approximately 5 times more potent than FT671, induces apoptosis, and exhibits a synergistic effect with mTOR inhibitors.

Molecular Formula

C29H32N4O4

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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