YCH2823
Product Specifications
Target
Apoptosis, DUB
Related Pathways
Cell Cycle/Checkpoint, Apoptosis, DNA Damage/DNA Repair, Ubiquitination
Bioactivity
YCH2823 is an inhibitor of USP7 (IC50= 49.6 nM; Kd= 0.117 μM) and demonstrates significant efficacy in suppressing both wild-type TP53 tumors and mutated tumors. It is approximately 5 times more potent than FT671, induces apoptosis, and exhibits a synergistic effect with mTOR inhibitors.
Molecular Formula
C29H32N4O4
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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