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Anticancer agent 201

Product Specifications

Target

Apoptosis|||Caspase|||PARP|||Bcl-2 Family

Related Pathways

Chromatin/Epigenetic|||DNA Damage/DNA Repair|||Apoptosis|||Proteases/Proteasome

Bioactivity

Anticanceragent 201 (Compound 2f) exhibits IC50 values in the low micromolar range across various tumor cell lines. It demonstrates high in vitro cytotoxicity against CCRF-CEM cells by inducing apoptosis through the activation of caspase-3 in the mitochondrial intrinsic pathway, cleavage of PARP, and reduced expression of Bcl-2 and Bcl-XL proteins. Anticanceragent 201 can be utilized in cancer research.

Molecular Formula

C34H49F3O4

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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