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A2AR/A2BR antagonist 1

Product Specifications

Target

Adenosine Receptor

Related Pathways

Neuroscience|||GPCR/G Protein

Bioactivity

A2AR/A2BR antagonist 1 (compound 7ai) acts as a dual antagonist to A2AR and A2BR with IC50 values of 11.2 nM and 6.4 nM, respectively. Additionally, A2AR/A2BR antagonist 1 enhances T cell-mediated cancer cell death.

Molecular Formula

C24H17N9

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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