TRPV1 antagonist 6
Product Specifications
Target
TRP/TRPV Channel
Related Pathways
Membrane transporter/Ion channel
Bioactivity
TRPV1 antagonist 6 (compound 51) is a modality-selective TRPV1 antagonist that exhibits antagonistic activity against capsaicin activation with an IC50 of 2.85 nM and demonstrates an inhibition rate of 28.48% against proton activation at a concentration of 3 μM.
Molecular Formula
C26H28ClN5O3
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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