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Dyrk1A-IN-7

Product Specifications

Target

DYRK

Related Pathways

Cell Cycle/Checkpoint, Tyrosine Kinase/Adaptors

Bioactivity

Dyrk1A-IN-7 (Compound 29) is a selective DYRK1A kinase inhibitor with notable kinase selectivity, exhibiting an IC50 value of 28 nM for DYRK1A and a Kd of 17.5 nM for CLK2. This selective inhibitor is applicable in research related to cancer, type II diabetes, and neurological disorders.

Molecular Formula

C19H13F3N4O

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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