GPR183 antagonist-3
Product Specifications
Target
EBI2/GPR183
Related Pathways
GPCR/G Protein
Bioactivity
GPR183 antagonist-3 (compound 33) is an orally active GPR183 antagonist with an IC50 value of 8.7 μM. It demonstrates significant in vitro anti-migration and anti-inflammatory activity in monocytes and can alleviate pathological symptoms in experimental colitis induced by dextran sulfate sodium.
Molecular Formula
C21H19BrN4O2S
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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