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C5aR1 antagonist 1

Product Specifications

Target

Complement System

Related Pathways

Immunology/Inflammation

Bioactivity

C5aR1 antagonist 1 (compound 7e) is an orally active C5a receptor antagonist. It demonstrates efficacy in both DISCO and migration assays, with IC50 values of 38 nM and 17 nM, respectively. This compound is useful for research in both acute and chronic inflammatory diseases.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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