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PPAR? agonist 10

Product Specifications

Target

PPAR

Related Pathways

DNA Damage/DNA Repair|||Metabolism

Bioactivity

PPAR? agonist10 (compound 7) is an orally active, selective partial agonist of PPAR?, with EC50 values of 0.053 ?M for hPPAR? (LBD) -GAL4 and 0.30 µM for mPPAR?. In transactivation assays, it acts as a partial PPAR? agonist but fully stimulates muscle cell free fatty acid oxidation both in vitro and in vivo. PPAR? agonist10 can be utilized for dyslipidemia research.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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