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PPARδ agonist 10

Product Specifications

Target

PPAR

Related Pathways

DNA Damage/DNA Repair, Metabolism

Bioactivity

PPARδ agonist10 (compound 7) is an orally active, selective partial agonist of PPARδ, with EC50 values of 0.053 μM for hPPARδ (LBD) -GAL4 and 0.30 μM for mPPARδ. In transactivation assays, it acts as a partial PPARδ agonist but fully stimulates muscle cell free fatty acid oxidation both in vitro and in vivo. PPARδ agonist10 can be utilized for dyslipidemia research.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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