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MAGL-IN-13

Product Specifications

Target

MAGL|||Calcium Channel

Related Pathways

Membrane transporter/Ion channel|||Metabolism

Bioactivity

MAGL-IN-13 (compound (3R,4S) -5v) is a selective, irreversible MAGL inhibitor with IC50 values of 0.026 nM for mMAGL, 0.021 nM for hMAGL, and 0.24 nM for rMAGL. Additionally, MAGL-IN-13 is capable of crossing the blood-brain barrier.

Molecular Formula

C28H24FN5O4

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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