EGFR/ACK1-IN-1
Product Specifications
Target
EGFR, ACK1
Related Pathways
JAK/STAT signaling, Tyrosine Kinase/Adaptors, Angiogenesis
Bioactivity
EGFRT790M/L858R/ACK1-IN-1 (Compound 21a) is a dual inhibitor targeting EGFRT790M/L858R and ACK1 with IC50 values of 23 nM and 263 nM, respectively. This compound effectively inhibits cell proliferation and exhibits antitumor activity.
Molecular Formula
C22H20ClN7O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
More Discoveries
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