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Nav1.8-IN-6

Product Specifications

Target

Sodium Channel

Related Pathways

Membrane transporter/Ion channel

Bioactivity

Nav1.8-IN-6 (Compound 2j) is a novel pyridinone amide Nav1.8 channel inhibitor with IC50 values of 513.33 nM in the resting state and 471.81 nM in the partially activated state. Nav1.8-IN-6 also exhibits analgesic activity.

Molecular Formula

C19H17F6N3O2

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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