CI-988 hemihydrate
Product Specifications
Target
Cholecystokinin Receptor
Related Pathways
GPCR/G Protein
Bioactivity
CI-988 hemihydrate (PD134308) is a potent and selective orally active CCK2R (cholecystokinin 2 receptor) antagonist, with an IC50 of 1.7 nM for mouse cortical CCK2. It is over 1600 times more selective for CCK2 than for CCK1 receptors. CI-988 hemihydrate exhibits anxiolytic and antitumor properties.
Molecular Formula
C35H42N4O6.1/2H2O
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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