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WDR5-IN-8

Product Specifications

Target

JAK

Related Pathways

JAK/STAT signaling|||Tyrosine Kinase/Adaptors|||Angiogenesis|||Chromatin/Epigenetic|||Stem Cells

Bioactivity

WDR5-IN-8 is a WDR5 inhibitor with an IC50 value of 15.5 nM. It displays significant antiproliferative activity in two human acute leukemia cell lines and possesses antitumor properties.

Molecular Formula

C29H29ClN4O2

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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