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BHEPN

Product Specifications

Target

VEGFR

Related Pathways

Angiogenesis, Tyrosine Kinase/Adaptors

Bioactivity

BHEPN is an inhibitor of vascular endothelial growth factor receptor-2 (VEGFR-2), exhibiting an inhibitory effect with an IC50 value of 0.320 μM. It also demonstrates significant cytotoxic activity against HepG2 and MCF-7 cancer cell lines, with IC50 values of 0.19 μM and 1.18 μM, respectively. BHEPN is applicable for cancer research.

Molecular Formula

C21H17BrN4O2

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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