σ1 Receptor/μ Opioid receptor modulator 2
Product Specifications
CAS Number
3009018-61-2
Target
Sigma receptor, Opioid Receptor
Related Pathways
Endocrinology/Hormones, Neuroscience, GPCR/G Protein
Bioactivity
Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM) . It demonstrates significant analgesic effects in various pain models.
Smiles
O=C(N(C1=NC=CC=C1)CC(N2CCC(C=3C=CC=CC3)CC2)CC)CC
Molecular Formula
C23H31N3O
Molecular Weight
365.51
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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