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T-1-DOCA

Product Specifications

Target

EGFR|||Apoptosis

Related Pathways

JAK/STAT signaling|||Apoptosis|||Angiogenesis|||Tyrosine Kinase/Adaptors

Bioactivity

T-1-DOCA is an EGFR inhibitor with IC50 values of 56.94 nM for EGFRWT and 269.01 nM for EGFRT790M. It has the capability to induce apoptosis (cellapoptosis) in HCT-116 cells.

Molecular Formula

C15H13Cl2N5O3

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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