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EGFR-IN-94

Product Specifications

Target

Apoptosis, VEGFR, EGFR

Related Pathways

Tyrosine Kinase/Adaptors, Angiogenesis, Apoptosis, JAK/STAT signaling

Bioactivity

EGFR-IN-94 (compound 5a) is an EGFR inhibitor with an IC50 of 0.086 μM. It exhibits IC50 values of 0.107 μM for VEGFR-2 and 2.52 μM for Topo II. In HepG-2 cells, EGFR-IN-94 induces apoptosis and causes cell cycle arrest at the S phase.

Molecular Formula

C19H17ClN8OS

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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