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AChE/BChE-IN-16

Product Specifications

Target

Cholinesterase (ChE) |||Reactive Oxygen Species

Related Pathways

NF-?B|||Metabolism|||Immunology/Inflammation|||Neuroscience

Bioactivity

AChE/BChE-IN-16 (compound C7) is a potent cholinesterase (ChE) inhibitor, exhibiting IC50 values of 30 nM for human acetylcholinesterase (hAChE) and 48 nM for human butyrylcholinesterase (hBuChE) . It demonstrates remarkable protective effects on PC12 cells against H2O2-induced apoptosis and effectively inhibits the production of reactive oxygen species (ROS) .

Molecular Formula

C33H34FN5O2

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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