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HL403

Product Specifications

Target

Src, Epigenetic Reader Domain

Related Pathways

Angiogenesis, Chromatin/Epigenetic, Tyrosine Kinase/Adaptors

Bioactivity

HL403 is a potent dual inhibitor targeting BRD4 and Src, with an IC50 value of 133 nM for BRD4 inhibition and 4.5 nM for Src inhibition. HL403 demonstrates anticancer activity.

Molecular Formula

C44H46Cl2N12O4S2

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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