What is the catalog number for SKLB-03220?

The catalog number for SKLB-03220 is T207811.

What sizes are available for SKLB-03220?

SKLB-03220 is available in the following size(s): 1 mg, 5 mg, 10 mg, 25 mg, 50 mg.

How many pack sizes does SKLB-03220 come in?

SKLB-03220 is available in 5 different pack sizes.

Is SKLB-03220 in stock?

SKLB-03220 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures SKLB-03220?

SKLB-03220 is manufactured by Molfinity.

What is the estimated delivery time for SKLB-03220?

Estimated delivery time for SKLB-03220 is approximately 10 business day(s), depending on your location.

SKLB-03220

Product Specifications

CAS Number

2852050-29-2

Target

Histone Methyltransferase

Related Pathways

Chromatin/Epigenetic

Purity

0.97016

Bioactivity

SKLB-03220 is an orally bioavailable covalent inhibitor targeting the histone methyltransferase EZH2, an established oncology drug target involved in epigenetic regulation. SKLB-03220 is structurally based on the clinically approved EZH2 inhibitor tazemetostat and demonstrates the ability to abolish epigenetic H3K27me3 marks, thereby altering chromatin state and transcriptional activity. SKLB-03220 represents a potent small-molecule tool for cancer epigenetics research.