SKLB-03220
Product Specifications
CAS Number
2852050-29-2
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9702
Bioactivity
SKLB-03220 is an orally bioavailable covalent inhibitor targeting the histone methyltransferase EZH2, an established oncology drug target involved in epigenetic regulation. SKLB-03220 is structurally based on the clinically approved EZH2 inhibitor tazemetostat and demonstrates the ability to abolish epigenetic H3K27me3 marks, thereby altering chromatin state and transcriptional activity. SKLB-03220 represents a potent small-molecule tool for cancer epigenetics research.
Smiles
O=C(C=C)NC1=CC=C(C(=C1)C=2C=C(C(=O)NCC=3C(=O)NC(=CC3C)C)C(=C(C2)N(CC)C4CCOCC4)C)C
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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