CB1R Allosteric modulator 5
Product Specifications
CAS Number
3019958-44-9
Target
Cannabinoid Receptor
Related Pathways
GPCR/G Protein
Bioactivity
CB1R Allosteric modulator 5 (compound 3) is a selective allosteric modulator of cannabinoid receptor type 1 (Cannabinoid receptor type 1) that can cross the blood-brain barrier, with a pIC0 value of 6.89. It reduces cue-induced reinstatement of cocaine-seeking behavior and cocaine-induced behavioral sensitization without altering motor activity.
Smiles
O=C1C(=O)C(NCCC=2C=CC=C(Cl)C2)=C1NC3=CC=C(Cl)C=C3
Molecular Formula
C18H14Cl2N2O2
Molecular Weight
361.22
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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