FGFR-IN-20
Product Specifications
Target
FGFR
Related Pathways
Tyrosine Kinase/Adaptors, Angiogenesis
Bioactivity
Glu-IN-1 (compound AF1) is a covalent inhibitor selectively targeting FGFR2, with an IC50 of 1.6 μM. It covalently modifies Glu489 in FGFR2.
Molecular Formula
C36H43N5O3
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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