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FGFR-IN-20

Product Specifications

Target

FGFR

Related Pathways

Tyrosine Kinase/Adaptors, Angiogenesis

Bioactivity

Glu-IN-1 (compound AF1) is a covalent inhibitor selectively targeting FGFR2, with an IC50 of 1.6 μM. It covalently modifies Glu489 in FGFR2.

Molecular Formula

C36H43N5O3

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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