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EGFR-IN-87 hydrochloride

Product Specifications

Target

EGFR

Related Pathways

JAK/STAT signaling|||Angiogenesis|||Tyrosine Kinase/Adaptors

Bioactivity

EGFR-IN-87 (Compound Example 2) hydrochloride is an EGFR tyrosine kinase inhibitor. It has IC50 values of 3.1 nM, 1.3 nM, and 7.1 nM for EGFR_d746-750, EGFR_L858R/T790, and EGFR_WT, respectively, in A431 cells. EGFR-IN-87 hydrochloride is useful for cancer research.

Molecular Formula

C28H34ClN7O2

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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