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PLA2-IN-1

Product Specifications

Target

Phospholipase

Related Pathways

Metabolism

Bioactivity

PLA2-IN-1 (Compound 7) is a potent and selective inhibitor of phospholipase A (PLA2) with an IC50 value of 1 nM. It effectively inhibits PLA2-induced coagulation disorders in vitro and shows potential for use as an antidote for snake bites caused by cobra venom.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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2- (2- (2,5-Dioxo-2,5-dihydro-1H-pyrrol-1-yl) ethoxy) ethyl ((S) -1- (((S) -1- ((4- (hydroxymethyl) phenyl) amino) -1-oxo-5-ureidopentan-2-yl) amino) -3-methyl-1-oxobutan-2-yl) carbamate
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