EN1441
Product Specifications
CAS Number
2196448-47-0
Target
Androgen Receptor
Related Pathways
Endocrinology/Hormones
Bioactivity
EN1441 is a covalent degrader that targets the androgen receptor (AR) with an EC50 value of 4.2 μM, as well as its truncated variant AR-V7. It selectively and effectively degrades AR and AR-V7 in androgen-independent prostate cancer cells. EN1441 holds potential for research into androgen-independent prostate cancer.
Smiles
O=C(C=C)N1C2=CC(Cl)=CC=C2NC(=O)C1(C)C
Molecular Formula
C13H13ClN2O2
Molecular Weight
264.708
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
132862-HRP 100 µL
RSF1 (Remodeling and Spacing Factor 1, Rsf-1, HBV pX-associated Protein 8, Hepatitis B Virus X-associated Protein, p325 Subunit of RSF Chromatin-remodeling Complex, HBXAP, XAP8) (HRP)
Sign In for Pricing
View Details 446171-01 5 mg
Des (4-methylcyclohexyl) carbamoyl N-Methoxycarbonyl-N-methyl ortho-Glimepiride
Sign In for Pricing
View Details 446171-02 10 mg
Des (4-methylcyclohexyl) carbamoyl N-Methoxycarbonyl-N-methyl ortho-Glimepiride
Sign In for Pricing
View Details 
orb2906507-01 20 µg
Recombinant Human Olfactory receptor 51I2 (OR51I2)
Sign In for Pricing
View Details