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PDE4D inhibitor 1

Product Specifications

Target

PDE|||CXCR|||Interleukin|||TNF

Related Pathways

GPCR/G Protein|||Metabolism|||Autophagy|||Immunology/Inflammation|||Apoptosis

Bioactivity

PDE4-IN-1 is a PDE4 inhibitor characterized by high potency (IC50: 8.6 nM) and superior selectivity over other PDE subtypes. This compound inhibits the release of inflammatory cytokines and chemokines. Additionally, PDE4-IN-1 significantly restores the damaged cAMP-CREB signaling pathway, inhibits proliferation, and promotes differentiation to reverse psoriasis formation.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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