HRG038
Product Specifications
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Bioactivity
HRG038 is a selective covalent BRD4 degrader. It binds covalently to the E3 ubiquitin ligase CUL4 DCAF16, recruiting it to BRD4, which results in BRD4 ubiquitination and subsequent proteasomal degradation. HRG038 holds potential for cancer research.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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