MRS7799
Product Specifications
CAS Number
224040-19-1
Target
Adenosine Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Bioactivity
MRS7799 is a selective A3 Adenosine Receptor antagonist with Kd values of 0.55 nM for humans, 3.74 nM for mice, and 2.80 nM for rats. MRS7799 can be utilized in research related to neurodegenerative diseases, cancer, cardiac and cerebral ischemia, and autoimmune inflammatory diseases.
Smiles
O=C(NC1=NC(C=2C=C(C=C(C2)C)C)=C(S1)C=3C=CN=CC3)C=4C=NC=CC4
Molecular Formula
C22H18N4OS
Molecular Weight
386.47
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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