Cebranopadol hemicitrate
Product Specifications
CAS Number
863513-92-2
Target
Opioid Receptor
Related Pathways
Neuroscience|||GPCR/G Protein|||Endocrinology/Hormones
Bioactivity
Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and ?-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.
Smiles
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Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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