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TO-1187

Product Specifications

Target

PROTACs|||HDAC

Related Pathways

DNA Damage/DNA Repair|||PROTAC|||Chromatin/Epigenetic

Bioactivity

TO-1187 is a selective HDAC6 PROTAC degrader with a DC50 of 5.81 nM. It enhances the ubiquitination and subsequent degradation of HDAC6, making it useful for research in hematological malignancies and solid tumors.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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