What is the catalog number for PPARα agonist 5?

The catalog number for PPARα agonist 5 is T206549.

What sizes are available for PPARα agonist 5?

PPARα agonist 5 is available in the following size(s): 10 mg, 50 mg.

How many pack sizes does PPARα agonist 5 come in?

PPARα agonist 5 is available in 2 different pack sizes.

Is PPARα agonist 5 in stock?

PPARα agonist 5 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures PPARα agonist 5?

PPARα agonist 5 is manufactured by Molfinity.

What is the estimated delivery time for PPARα agonist 5?

Estimated delivery time for PPARα agonist 5 is approximately 10 business day(s), depending on your location.

PPARα agonist 5

Product Specifications

Target

Phosphatase, PPAR

Related Pathways

DNA Damage/DNA Repair, Metabolism

Bioactivity

PPARα agonist5 is an orally active, selective partial agonist of PPARα with an EC50 of 3 nM. It reduces lipid accumulation and upregulates PPARα target genes, exhibiting anti-hepatic steatosis properties. Additionally, PPARα agonist5 demonstrates significant lipid-lowering and glucose-lowering effects through partial PPARγ agonist activity and mild inhibition of protein tyrosine phosphatase 1B (PTP1B) with an IC50 of 79.1 μM. It has favorable safety and is applicable in the study of dyslipidemia in type 2 diabetes.