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Anticonvulsant agent 10

Product Specifications

Target

Nrf2

Related Pathways

Immunology/Inflammation

Bioactivity

Anticonvulsant agent 10 (Compound 6d) is an inhibitor targeting the Keap1-Nrf2 interaction, with a strong activity showing an ED50 of 0.04 mmol/kg. By inhibiting the Keap1-Nrf2 binding, it activates the Nrf2/ARE pathway, providing anticonvulsant and neuroprotective effects, making it useful for research in epilepsy and neuroprotection.

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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