CB1R agonist 1
Product Specifications
Target
Cannabinoid Receptor
Related Pathways
GPCR/G Protein
Bioactivity
CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.
Smiles
CC1=CC(C(N[C@@](C(OC)=O)(C)C2=CC=CS2)=O)=NN1C3=CC(C(F)(F)F)=CC=C3
Molecular Formula
C20H18F3N3O3S
Molecular Weight
437.435
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Product Datasheet
https://www.targetmol.com/attachment/DataSheet/347062797269467172/T206337
Available Sizes
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