Darlifarnib
Product Specifications
CAS Number
2939824-30-1
Target
Transferase
Related Pathways
Metabolism
Bioactivity
Darlifarnib (Compound (S) -058) is an inhibitor of farnesyl transferase and geranylgeranyltransferase, with IC50 values of ≤ 10 nM and > 1000 nM, respectively. It exhibits high metabolic stability in human and mouse liver microsomes, with a half-life of over 100 minutes.
Smiles
N#CC=1N=C2C=CC3=CC2=C(C1)C=4C=CC=C(OCC5=CC(=CC=C5C#N)C3(N)C6=CN=CN6C)C4
Molecular Formula
C29H20N6O
Molecular Weight
468.509
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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