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NNRT-IN-6

Product Specifications

Target

Reverse Transcriptase, HIV Protease

Related Pathways

Proteases/Proteasome, Microbiology/Virology

Bioactivity

NNRT-IN-6 (Compound 13a) is a non-nucleoside reverse transcriptase inhibitor (NNRT) used to inhibit HIV-1 reverse transcriptase (HIV-1RT), with an IC50 of 0.41 μM. It effectively suppresses both wild-type HIV-1 and mutants L100I, K103N, Y181C, Y188L, E138K, F227L/V106A, and RES056, with an EC50 range of 6.2-250 nM.

Molecular Formula

C32H31N9O3S

Molecular Weight

621.71

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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