H3R antagonist 5
Product Specifications
CAS Number
879368-27-1
Target
Histamine Receptor
Related Pathways
Neuroscience, Immunology/Inflammation, GPCR/G Protein
Bioactivity
H3R antagonist 5 (Compound 1b) is a selective inverse agonist of the histamine H3 receptor that can penetrate the blood-brain barrier, with an IC50 of 0.54 nM. It is applicable for research related to the central nervous system.
Smiles
O=C1O[C@]2(C=3C1=CC(OC)=CC3)CC[C@@H](C(N(CCN4CCCCC4)C)=O)CC2
Molecular Formula
C23H32N2O4
Molecular Weight
400.511
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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