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OA-Br-1

Product Specifications

Target

Apoptosis|||Phosphatase

Related Pathways

Apoptosis|||Metabolism

Bioactivity

OA-Br-1 is an orally active, selective inhibitor of PTP1B with an IC50 value of 7.08 ?M. It induces apoptosis and exhibits broad-spectrum anti-cancer cell proliferation activity. OA-Br-1 exerts anti-breast cancer effects both in vitro and in vivo through the PTP1B/PI3K/AKT signaling pathway.

Molecular Formula

C43H70BrNO8

Molecular Weight

808.92

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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