C-Met/Axl-IN-1
Product Specifications
Target
Apoptosis, c-Met/HGFR, TAM Receptor
Related Pathways
Apoptosis, Tyrosine Kinase/Adaptors
Bioactivity
C-Met/Axl-IN-1 (Compound 22a) is an oral, selective type II c-Met/Axl inhibitor with IC50 values of 1 nM and 10 nM, respectively. It effectively suppresses tumor cell proliferation, induces cell cycle arrest, and apoptosis (apoptosis), showcasing potent anti-tumor activity.
Molecular Formula
C25H18F2N6O2
Molecular Weight
472.45
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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