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PDE7A-IN-1

Product Specifications

Target

PDE

Related Pathways

Metabolism

Bioactivity

PDE7A-IN-1 (Compound 26) is an orally active PDE7A inhibitor with an IC50 value of 3.7 nM. By inhibiting sclerostin, PDE7A-IN-1 significantly enhances bone mineral density, making it suitable for studies on osteoporosis and related bone metabolic disorders.

Molecular Formula

C25H26ClN5O2

Molecular Weight

463.96

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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