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KOR agonist 5

Product Specifications

Target

Opioid Receptor

Related Pathways

Neuroscience|||Endocrinology/Hormones|||GPCR/G Protein

Bioactivity

KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD) .

Molecular Formula

C38H38N2O5

Molecular Weight

602.72

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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