KOR agonist 5
Product Specifications
Target
Opioid Receptor
Related Pathways
Neuroscience|||Endocrinology/Hormones|||GPCR/G Protein
Bioactivity
KOR agonist 5 (Compound 10a) is both a KOR/MOR modulator, exhibiting agonistic effects on KOR and antagonistic effects on MOR. It effectively blocks morphine-induced antinociception and gastrointestinal motility inhibition. KOR agonist 5 is applicable in research related to substance use disorder (SUD) .
Molecular Formula
C38H38N2O5
Molecular Weight
602.72
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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