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ErSO-TFPy

Product Specifications

CAS Number

3035547-78-2

Target

Sodium Channel

Related Pathways

Membrane transporter/Ion channel

Bioactivity

ErSO-TFPy activates the sodium ion channel TRPM4, resulting in an imbalance of intracellular calcium and sodium ions. It exhibits low nanomolar-level cytotoxicity (IC50 = 5-25 nM) by inducing necrosis in ER?+ breast cancer cell lines. Additionally, ErSO-TFPy shows antitumor activity in mouse models.

Smiles

O=C1[C@@](C=2C(N1)=C(C(F)(F)F)C=CC2)(N3CC(F)(F)C(F)(F)C3)C4=CC=C(O)C=C4

Molecular Formula

C19H13F7N2O2

Molecular Weight

434.307

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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