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Famlasertib

Product Specifications

CAS Number

2375591-69-6

Target

MAPK

Related Pathways

MAPK

Bioactivity

Famlasertib is a potent inhibitor of the mitogen-activated protein kinase kinase kinase kinase (MAP4K) family, capable of penetrating the brain. It exhibits an IC50 value of 0.3 nM for HGK (MAP4K4) and 23.7 nM for MLK3.

Smiles

ClC1=CC=CC(=C1)C2=CNC3=NC=C(C=C32)C=4C=CC(=CC4)CN5CCN(CCO)CC5

Molecular Formula

C26H27ClN4O

Molecular Weight

446.972

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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