What is the catalog number for HDAC3/BRD4-IN-1?

The catalog number for HDAC3/BRD4-IN-1 is T205214.

What sizes are available for HDAC3/BRD4-IN-1?

HDAC3/BRD4-IN-1 is available in the following size(s): 10 mg, 50 mg.

How many pack sizes does HDAC3/BRD4-IN-1 come in?

HDAC3/BRD4-IN-1 is available in 2 different pack sizes.

Is HDAC3/BRD4-IN-1 in stock?

HDAC3/BRD4-IN-1 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures HDAC3/BRD4-IN-1?

HDAC3/BRD4-IN-1 is manufactured by Molfinity.

What is the estimated delivery time for HDAC3/BRD4-IN-1?

Estimated delivery time for HDAC3/BRD4-IN-1 is approximately 10 business day(s), depending on your location.

HDAC3/BRD4-IN-1

Product Specifications

Target

Epigenetic Reader Domain, HDAC

Related Pathways

DNA Damage/DNA Repair, Chromatin/Epigenetic

Bioactivity

HDAC3/BRD4-IN-1 (compound 26n) is an inhibitor of HDAC3/BRD4, exhibiting an IC50 of 8 nM for HDAC3, while its IC50 values for HDAC1 and HDAC2 are 220 nM and 120 nM, respectively. It displays anti-tumor and anti-proliferative effects by upregulating Ac-H3 and downregulating c-Myc. The half-life of HDAC3/BRD4-IN-1 in human liver microsomes is 29.36 minutes.