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PIKfyve-IN-4

Product Specifications

Target

PI3K

Related Pathways

PI3K/Akt/mTOR signaling

Bioactivity

PIKfyve-IN-4 (Compound 40) is an orally active and selective phosphatidylinositol-3-phosphate 5-kinase (PIKfyve) inhibitor, with an IC50 of 0.60 nM, and demonstrates good systemic tolerability.

Molecular Formula

C16H14N4S

Molecular Weight

294.37

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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