Cav 3.1 blocker 1
Product Specifications
CAS Number
2158201-04-6
Target
Calcium Channel
Related Pathways
Metabolism, Membrane transporter/Ion channel
Bioactivity
Cav 3.1 blocker 1 (compound 12) is a T-type calcium channel inhibitor with an IC50 value of 160 nM for Cav3.1. It exhibits weaker inhibition on Cav 3.2 with an IC50 of 5000 nM and shows no inhibitory effect on Cav 3.3 and Cav 1.2 (IC50 > 10000 nM) .
Smiles
O=C(NCC=1C=CC=CC1OCC(F)(F)F)C2=NN(C3=CC=C(F)C=C3)C(C=4C=CC=CC4)=C2C(F)F
Molecular Formula
C26H19F6N3O2
Molecular Weight
519.438
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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